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LY2922470

Glpbio
Catalog No:GC36507-10mM (in 1mL DMSO) CAS No.:1423018-12-5 MDLNo: Brand:Glpbio purity: 特性: Purpose:LY2922470 是一种有效、选择性的,口服有效的 GPR40 激动剂,作用于 人 GPR40、小鼠 GPR40、大鼠 GPR40 的 EC50 值分别为 7 nM、1 nM、3 nM。LY2922470 可降低血糖水平,同时显著增加胰岛素和 GLP-1,具有治疗 2 型糖尿病 (T2DM) 的潜力。DMSO: ≥ 125 mg/mL (262.83 mM)
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